Top   >   Back   >   学術論文・プロシーディングス・著作 の検索結果 168 件中 130 件目

Golgi retention and oncogenic KIT signaling via PLCγ2-PKD2-PI4KIIIβ activation in gastrointestinal stromal tumor cells
[ 全著者名 ] Yuuki OBATA, Kazuo KUROKAWA, Takuro TOJIMA, Miyuki NATSUME, Isamu SHIINA, Tsuyoshi TAKAHASHI, Ryo ABE, Akihiko NAKANO, Toshirou NISHIDA
[ 掲載誌名 ] Cell Reports
[ 掲載年月 ] 2023年 9月
[ 著作区分 ] レフェリー付学術論文(外国語)
First Total Synthesis of Tanzawaic Acid B
[ 全著者名 ] Takatsugu MURATA, Hisazumi TSUTSUI, Takumi YOSHIDA, Hirokazu KUBOTA, Shintaro HIRAISHI, Hiyo NATSUKAWA, Yuki SUZUKI, Daiki HIRAGA, Takahiro MORI, Yutaro MAEKAWA, Satoru TATEYAMA, Kiyotaka TOYOYAMA, Keiichi ITO, Kyohei SUZUKI, Keita YONEKURA, Natsumi SHIBATA, Teruyuki SATO, Yasutaka TASAKI, Takehiko INOHANA, Atsuhiro TAKANO, Naoki EGASHIRA, Masaki HONDA, Yuma UMEZAKI, Isamu SHIINA
[ 掲載誌名 ] ACS Omega
[ 掲載年月 ] 2023年 7月
[ 著作区分 ] レフェリー付学術論文(外国語)
FLT3-ITD Transduces Autonomous Growth Signals during Its Biosynthetic Trafficking in Acute Myelogenous Leukemia Cells
[ 全著者名 ] Kouhei YAMAWAKI, Isamu SHIINA, Takatsugu MURATA, Satoru TATEYAMA, Yutarou MAEKAWA, Mariko NIWA, Motoyuki SHIMONAKA, Koji OKAMOTO, Toshihiro SUZUKI, Toshirou NISHIDA, Ryo ABE, Yuuki OBATA
[ 掲載誌名 ] Scientific Reports
[ 掲載年月 ] 2021年 11月
[ 著作区分 ] レフェリー付学術論文(外国語)
BRAP2 Inhibits the Ras/Raf/MEK and PI3K/Akt Pathways in Leukemia Cells, Thereby Inducing Apoptosis and Inhibiting Cell Growth
[ 全著者名 ] Hiroharu SAKAI, Isamu SHIINA, Takahisa SHINOMIYA, Yukitoshi NAGAHARA
[ 掲載誌名 ] Experimental and Therapeutic Medicine
[ 掲載年月 ] 2021年 3月
[ 著作区分 ] レフェリー付学術論文(外国語)
4-(Dimethylamino)pyridine N-Oxide-Catalyzed Macrolactamization Using 2-Methyl-6-nitrobenzoic Anhydride in the Synthesis of the Depsipeptidic Analogue of FE399
[ 全著者名 ] Takayuki TONOI, Takehiko INOHANA, Ryo KAWAHARA, Teruyuki SATO, Miyuki IKEDA, Miku AKUTSU, Takatsugu MURATA, Isamu SHIINA
[ 掲載誌名 ] ACS Omega
[ 掲載年月 ] 2021年 2月
[ 著作区分 ] レフェリー付学術論文(外国語)
Total Synthesis of the Antitumor Depsipeptide FE399 and Its S-Benzyl Derivative: A Macrolactamization Approach
[ 全著者名 ] Takayuki TONOI, Miyuki IKEDA, Teruyuki SATO, Takehiko INOHANA, Ryo KAWAHARA, Takatsugu MURATA, Isamu SHIINA
[ 掲載誌名 ] EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
[ 掲載年月 ] 2020年 8月
[ 著作区分 ] レフェリー付学術論文(外国語)
Kinetic Resolution of Racemic 2-Hydroxyarylketones by Asymmetric Esterification: Investigation of the Influence of the Co-Base on the Selectivity
[ 全著者名 ] Takatsugu MURATA, Kengo FUTAMI, Ryo ISHIKAWA, Keisuke ONO, Kenya NAKATA, Isamu SHIINA
[ 掲載誌名 ] ASIAN J ORG CHEM
[ 掲載年月 ] 2020年 2月
[ 著作区分 ] レフェリー付学術論文(外国語)
Total Synthesis and Antimicrobial Evaluation of 23-Demethyleushearilide and Extensive Antimicrobial Evaluation of All Synthetic Stereoisomers of (16Z,20E)-Eushearilide and (16E,20E)-Eushearilide
[ 全著者名 ] Takayuki TONOI, Takehiko INOHANA, Teruyuki SATO, Yuuki NODA, Miyuki IKEDA, Miku AKUTSU, Takatsugu MURATA, Yutaro MAEKAWA, Anna TANAKA, Rio SEKI, Misako OHKUSU, Katsuhiko KAMEI, Naruhiko ISHIWADA, Isamu SHIINA
[ 掲載誌名 ] MOLECULES
[ 掲載年月 ] 2019年 9月
[ 著作区分 ] レフェリー付学術論文(外国語)
N822K- or V560G-mutated KIT activation preferentially occurs in lipid rafts of the Golgi apparatus in leukemia cells
[ 全著者名 ] Yuuki OBATA, Yasushi HARA, Isamu SHIINA, Takatsugu MURATA, Yasutaka TASAKI, Kyohei SUZUKI, Keiichi ITO, Shou TSUGAWA, Kouhei YAMAWAKI, Tsuyoshi TAKAHASHI, Koji OKAMOTO, Toshirou NISHIDA, Ryo ABE
[ 掲載誌名 ] CELL COMMUN SIGNAL
[ 掲載年月 ] 2019年 9月
[ 著作区分 ] レフェリー付学術論文(外国語)
DIASTEREO–/ENANTIOSELECTIVE DIELS–ALDER SYNTHESIS OF 14β-HYDROXYSTEROID SCAFFOLDS: A COMBINED EXPERIMENTAL AND DFT STUDY
[ 全著者名 ] Clovis Peter, Philippe Geoffroy, Takatsugu Murata, Takayuki Tonoi, Isamu Shiina, Michel Miesch
[ 掲載誌名 ] HETEROCYCLES
[ 掲載年月 ] 2019年 6月
[ 著作区分 ] レフェリー付学術論文(外国語)
Novel Ridaifen-B Structure Analog Induces Apoptosis and Autophagy Depending on Pyrrolidine Side Chain
[ 全著者名 ] Takumi Iwasawa, Takahisa Shinomiya, Nozomi Ota, Natsumi Shibata, Kenya Nakata, Isamu Shiina, Yukitoshi Nagahara
[ 掲載誌名 ] BIOLOGICAL & PHARMACEUTICAL BULLETIN
[ 掲載年月 ] 2019年 3月
[ 著作区分 ] レフェリー付学術論文(外国語)
Total Synthesis of Violaceoid A and (−)- and (+)-Violaceoid B
[ 全著者名 ] Takatsugu MURATA, Teppei KUBOKI, Ryo ISHIKAWA, Takahiro SAITO, Shotaro TAGUCHI, Kazuma TAKEUCHI, Emiko HATANO, Motoyuki SHIMONAKA, Isamu SHIINA
[ 掲載誌名 ] JOURNAL OF NATURAL PRODUCTS
[ 掲載年月 ] 2018年 11月
[ 著作区分 ] レフェリー付学術論文(外国語)
Kinetic Resolution of Racemic 2-Hydroxyamides Using a Diphenylacetyl Component as an Acyl Source and a Chiral Acyl-Transfer Catalyst
[ 全著者名 ] Takatsugu MURATA, Tatsuya KAWANISHI, Akihiro SEKIGUCHI, Ryo ISHIKAWA, Keisuke ONO, Kenya NAKATA, Isamu SHIINA
[ 掲載誌名 ] MOLECULES
[ 掲載年月 ] 2018年 8月
[ 著作区分 ] レフェリー付学術論文(外国語)
Total Synthesis and Antimicrobial Activities of All Stereoisomers of (16Z,20E)‐Eushearilide and (16E,20E)‐Eushearilide
[ 全著者名 ] Takayuki TONOI, Takehiko INOHANA, Teruyuki SATO, Tomoki YOSHIDA, Isamu SHIINA
[ 掲載誌名 ] JOURNAL OF ORGANIC CHEMISTRY
[ 掲載年月 ] 2018年 8月
[ 著作区分 ] レフェリー付学術論文(外国語)
Anti‐proliferative Effect of Ridaifen‐B on Hepatoma Cells
[ 全著者名 ] Go HASEGAWA, Kotomi AKATSUKA, Keita HIRUMA, Kayako SUDA, Yumiko YOKOE, Akihito MIZUSAWA, Nozomi OTA, Natsumi SHIBATA, Kaho TSUCHIYA, Moyuru HAYASHI, Isamu SHIINA, Motoyuki SHIMONAKA
[ 掲載誌名 ] Biomedical Reports
[ 掲載年月 ] 2018年 6月
[ 著作区分 ] レフェリー付学術論文(外国語)
Asymmetric Total Synthesis of (+)-Coprophilin
[ 全著者名 ] Isamu SHIINA, Yuma UMEZAKI, Takatsugu MURATA, Kyohei SUZUKI, Takayuki TONOI
[ 掲載誌名 ] SYNTHESIS-STUTTGART
[ 掲載年月 ] 2018年 3月
[ 著作区分 ] レフェリー付学術論文(外国語)
Ridaifen-F Conjugated with Cell-Penetrating Peptides Inhibits Intracellular Proteasome Activities and Induces Drug-Resistant Cell Death
[ 全著者名 ] Makoto Tanaka, Yunhao Zhu, Masafumi Shionyu, Nozomi Ota, Natsumi Shibata, Chihiro Watanabe, Akihito Mizusawa, Ryuzo Sasaki, Tamio Mizukami, Isamu Shiina, Makoto Hasegawa
[ 掲載誌名 ] EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
[ 掲載年月 ] 2018年 2月
[ 著作区分 ] レフェリー付学術論文(外国語)
Oncogenic Kit signalling on the Golgi is suppressed by blocking secretory trafficking with M-COPA in gastrointestinal stromal tumours
[ 全著者名 ] Yuuki Obata, Keita Horikawa, Isamu Shiina, Tsuyoshi Takahashi, Takatsugu Murata, Yasutaka Tasaki, Kyohei Suzuki, Keita Yonekura, Hiroyasu Esumi, Toshirou Nishida, Ryo Abe
[ 掲載誌名 ] CANCER LETTERS
[ 掲載年月 ] 2018年 2月
[ 著作区分 ] レフェリー付学術論文(外国語)
Targeting the Golgi apparatus to overcome acquired resistance of non-small cell lung cancer cells to EGFR tyrosine kinase inhibitors
[ 全著者名 ] Yoshimi Ohashi, Mutsumi Okamura, Ryohei Katayama, Siyang Fang, Saki Tsutsui, Akinobu Akatsuka, Mingde Shan, Hyeong-Wook Choi, Naoya Fujita, Kentaro Yoshimatsu, Isamu Shiina, Takao Yamori, Shingo Dan
[ 掲載誌名 ] Oncotarget
[ 掲載年月 ] 2018年 1月
[ 著作区分 ] レフェリー付学術論文(外国語)
Family-wide Analysis of the Inhibition of Arf Guanine Nucleotide Exchange Factors with Small Molecules: Evidence of Unique Inhibitory Profiles
[ 全著者名 ] Sarah BENABDI, François PEUROIS, Agata NAWROTEK, Jahnavi CHIKIREDDY, Tatiana CAÑEQUE, Takao YAMORI, Isamu SHIINA, Yoshimi OHASHI, Shingo DAN, Raphaël RODRIGUEZ, Jacqueline CHERFILS, Mahel ZEGHOUF
[ 掲載誌名 ] BIOCHEMISTRY
[ 掲載年月 ] 2017年 9月
[ 著作区分 ] レフェリー付学術論文(外国語)
Asymmetric Total Synthesis of (−)-Astakolactin and Confirmation of Its Stereostructure
[ 全著者名 ] Takayuki TONOI, Yutaka YOSHINAGA, Moe FUJISHIRO, Keisuke MAMEDA, Takashi KATO, Kentaro SHIBAMOTO, Isamu SHIINA
[ 掲載誌名 ] JOURNAL OF NATURAL PRODUCTS
[ 掲載年月 ] 2017年 8月
[ 著作区分 ] レフェリー付学術論文(外国語)
Acylative Kinetic Resolution of Racemic Aromatic β-Hydroxy Esters Catalyzed by Chiral Nucleophilic N-(1-Arylethyl)benzoguanidines
[ 全著者名 ] Akira Yamada, Isamu SHIINA, and Kenya NAKATA
[ 掲載誌名 ] TETRAHEDRON-ASYMMETRY
[ 掲載年月 ] 2017年 4月
[ 著作区分 ] レフェリー付学術論文(外国語)
M-COPA Suppresses Endolysosomal Kit-Akt Oncogenic Signalling through Inhibiting the Secretory Pathway in Neoplastic Mast Cells
[ 全著者名 ] Yasushi Hara, Yuuki Obata, Keita Horikawa, Yasutaka Tasaki, Kyohei Suzuki, Takatsugu Murata, Isamu Shiina, and Ryo Abe
[ 掲載誌名 ] PLoS One
[ 掲載年月 ] 2017年 4月
[ 著作区分 ] レフェリー付学術論文(外国語)
EXPEDITIOUS SYNTHESIS OF CARBOXYLIC ESTERS AND HIGH-YIELDING MACROLACTONES USING TRIFLUOROMETHYL-SUBSTITUTED BENZOIC ANHYDRIDES WITH 4-(DIMETHYLAMINO)PYRIDINE: AN EVALUATION OF THE REACTIVITIES OF AROMATIC ACID ANHYDRIDES AS DEHYDRATION REAGENTS COMPARED WITH 2-METHYL-6-NITROBENZOIC ANHYDRIDE
[ 全著者名 ] Isamu SHIINA and Takayuki TONOI
[ 掲載誌名 ] HETEROCYCLES
[ 掲載年月 ] 2017年 2月
[ 著作区分 ] レフェリー付学術論文(外国語)
KINETIC RESOLUTION OF RACEMIC 2-HYDROXYACETALS BY ASYMMETRIC ESTERIFICATION USING A MIXED ANHYDRIDE PROTOCOL
[ 全著者名 ] Kenya Nakata, Eri Tokumaru, Takahiro Saitoh, Takayoshi Nakahara, Keisuke Ono, Takatsugu Murata, and Isamu Shiina
[ 掲載誌名 ] HETEROCYCLES
[ 掲載年月 ] 2016年 10月
[ 著作区分 ] レフェリー付学術論文(外国語)
Enantioselective Total Synthesis of Naturally Occurring Eushearilide and Evaluation of Its Antifungal Activity
[ 全著者名 ] Takayuki TONOI, Ryo KAWAHARA, Takehiko INOHANA, and Isamu SHIINA
[ 掲載誌名 ] JOURNAL OF ANTIBIOTICS
[ 掲載年月 ] 2016年 9月
[ 著作区分 ] レフェリー付学術論文(外国語)
M-COPA, a Novel Golgi System Disruptor, Suppresses Apoptosis Induced by Shiga Toxin
[ 全著者名 ] Takayuki HATTORI, Miho WATANABE-TAKAHASHI, Isamu SHIINA, Yoshimi OHASHI, Shingo DAN, Kiyotaka NISHIKAWA, Takao YAMORI, and Mikihiko NAITO
[ 掲載誌名 ] GENES TO CELLS
[ 掲載年月 ] 2016年 8月
[ 著作区分 ] レフェリー付学術論文(外国語)
M-COPA, a Golgi Disruptor, Inhibits Cell Surface Expression of MET Protein and Exhibits Antitumor Activity against MET-Addicted Gastric Cancers
[ 全著者名 ] Yoshimi OHASHI, Mutsumi OKAMURA, Asaka HIROSAWA, Naomi TAMAKI, Akinobu AKATSUKA, Kuo-Ming WU, Hyeong-Wook CHOI, Kentaro YOSHIMATSU, Isamu SHIINA, Takao YAMORI, and Shingo DAN
[ 掲載誌名 ] CANCER RESEARCH
[ 掲載年月 ] 2016年 7月
[ 著作区分 ] レフェリー付学術論文(外国語)
不斉エステル化反応を用いたキラル医薬品の合成―抗炎症剤および抗肥満薬の製造を例として― Synthesis of Chiral Pharmaceutical Drugs by Using Asymmetric Esterification―Application for the Production of Non-Steroidal Anti-Inflammatory Drugs; NSAIDs, and Tetrahydrolipstatin; THL―
[ 全著者名 ] 中田健也、殿井貴之、椎名 勇
[ 掲載誌名 ] 月刊ファインケミカル
[ 掲載年月 ] 2016年 2月
[ 著作区分 ] レフェリー付学術論文(日本語)
Nonenzymatic, Enantioconvergent Dynamic Kinetic Resolution (DKR) of Racemic 2-(1H-Pyrrol-1-yl)alkanoic Acids as α-Amino Acid Equivalents
[ 全著者名 ] Eri TOKUMARU, Atsushi TENGEIJI, Takayoshi NAKAHARA, and Isamu SHIINA
[ 掲載誌名 ] CHEMISTRY LETTERS
[ 掲載年月 ] 2015年 12月
[ 著作区分 ] レフェリー付学術論文(外国語)
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